A Step-Economical Multicomponent Synthesis of 3D-Shaped Aza-Diketopiperazines and Their Drug-like Chemical Space Analysis

Org. Biomol. Chem., 2016, Accepted ManuscriptDOI: 10.1039/C6OB01434H, PaperPierre-Michel Regenass, Stephanie Riche, Florent Peron, Didier Rognan, Marcel Hibert, Nicolas Girard, Dominique BonnetA rapid and atom economy multicomponent synthesis of complex aza-diketopiperazines (aza-DKPs) driven by Rh(I)-catalyzed hydroformylation of alkenylsemicarbazides is described.

Total Synthesis of Cananginone C and Structural Revision of Debilisone A

Org. Biomol. Chem., 2016, Accepted ManuscriptDOI: 10.1039/C6OB01671E, PaperTapan Kumar Kuilya, RAJIB KUMAR GOSWAMIA short, convergent and general strategy for stereoselective total synthesis of biologically active [small alpha]-substituted [gamma]-hydroxymethyl [gamma]-lactone based natural products cananginone C and debilisone A has been developed. The salient features...The content of this RSS Feed (c) The Royal Society of Chemistry

4,4?-Bismoschamine: Biomimetic Synthesis and Evidence to Support Structural Equivalency to Montamine

Org. Biomol. Chem., 2016, Accepted ManuscriptDOI: 10.1039/C6OB01685E, PaperKaitlin G. Henry, Lachlan Blair, Jonathan Sperry, Elizabeth Colby DavieThe dimeric natural product montamine was originally reported as two N-feruloylserotonin (moschamine) units linked by a nitrogen-nitrogen bond, but our recent synthesis of this symmetrical diacyl hydrazide structure revealed this...The content of this RSS Feed (c) The Royal Society of Chemistry

Total Synthesis of Mangiferin, Homomangiferin, and Neomangiferin

Org. Biomol. Chem., 2016, Accepted ManuscriptDOI: 10.1039/C6OB01622G, PaperXiong Wei, Danlin Liang, Qing Wang, Xiangbao Meng, Zhongjun LiTotal synthesis of mangiferin, homomangiferin, and neomangiferin, three C-glycosyl xanthone natural products with a wide spectrum of pharmacological effects, have been achieved starting from 2,3,4,6-tetra-O-benzyl-glucopyranose.

A Protecting Group-Free Synthesis of (-)-Hortonones A-C from the Inhoffen-Lythgoe Diol

Org. Biomol. Chem., 2016, Accepted ManuscriptDOI: 10.1039/C6OB01738J, PaperHovsep Stambulyan, Thomas MinehanA synthesis of hortonones A-C has been accomplished from Vitamin D2 via the Inhoffen-Lythgoe diol without the use of protective groups. Key steps in the syntheses include a TMS-diazomethane mediated...The content of this RSS Feed (c) The Royal Society of Chemistry

Traceless switch organocatalysis enables multiblock ring-opening copolymerizations of lactones, carbonate, and lactide: by one plus one and in one-pot

Polym. Chem., 2016, Accepted ManuscriptDOI: 10.1039/C6PY01107A, PaperXin Wang, Jiaqi Liu, Songquan Xu, Jiaxi Xu, Xianfu Pan, Jingjing Liu, Saide Cui, Zhenjiang Li, Kai GuoCatalytic ring-opening polymerization (ROP) of the three major types of cyclic monomers of lactides, lactones, and carbonates showed match and mismatch between the monomer and the catalyst.

Enhanced stability of conductive polyacetylene in ladder-like surface-grafted brushes

Polym. Chem., 2016, Accepted ManuscriptDOI: 10.1039/C6PY00977H, PaperMichal Szuwarzynski, Karol Wolski, Szczepan ZapotocznyFormation and characterization of polyacetylene-based brushes that exhibit exceptional long term stability in air is presented here. Polyacetylene, structurally the simplest conjugated polymer, exhibits the highest conductivity among them but...The content of this RSS Feed (c) The Royal Society of Chemistry

Synthesis and biomedical applications of fluorescent nanogels

Polym. Chem., 2016, Accepted ManuscriptDOI: 10.1039/C6PY01021K, Review ArticleWei Liu, Wensi Zhang, Xiaoqing Yu, Guanghua Zhang, Zhiqiang SuFluorescent nanogel is innovative biomedical material with hydroscopicity, degradability, responsiveness. It has attracted increasing attentions over the past years due to the unique fluorescence properties provided by different fluorophores.

Lipid droplet size and emulsification on postprandial glycemia, insulinemia and lipidemia

Food Funct., 2016, Accepted ManuscriptDOI: 10.1039/C6FO00897F, PaperKevin Wei Jie Tan, Lijuan Sun, Kelvin Kim Tha Goh, Henry JeyakumarPrevious studies have suggested that smaller lipid droplet size results in greater rate of lipolysis. However, acute health impacts of emulsification and small lipid droplet size is not well understood....The content of this RSS Feed (c) The Royal Society of Chemistry

Kinetically-Enhanced Polysul?de Redox Reactions by Nb2O5 Nanocrystal for High-Rate Lithium-Sulfur Battery

Energy Environ. Sci., 2016, Accepted ManuscriptDOI: 10.1039/C6EE01662F, PaperDonghui Long, Yingiqng Tao, Yanju Wei, Yu Liu, Jitong Wang, Wen M Qiao, Licheng LingTo combat the shuttle of soluble polysul?des, physical confinement approaches aiming to trap sulfur within porous hosts have been pursued, but their success towards capacity decay and kinetic sluggishness is...The content of this RSS Feed (c) The Royal Society of Chemistry

Amaysim completes AU$4m AusBBS acquisition

Amaysim has issued AU$1.5 million in shares and paid AU$1 million in cash to acquire AusBBS, and is due to pay an additional AU$1.5 million in shares in a year.

Turkey strikes IS and Kurdish positions in Syria ahead of offensive

Turkey bombards so-called Islamic State (IS) targets in northern Syria ahead of a ground offensive it is backing against the group.

?Victoria soon to make Uber legal

The Victorian government will introduce draft legislation this year as part of a two-year move to overhaul regulations governing the commercial passenger industry.

Tokyo Olympics 2020: 10 potential stars of the next Olympics

Who might shine at Tokyo 2020? Contenders include a cyclist who had a team-mate in tears and a sprinter out to match Usain Bolt.

Optus and Telstra compete on streaming inclusions

Optus is offering greater instances of unmetered streaming, while Telstra throws in more free subscriptions for streaming services in an effort to attract customers.

Mothers' pay lags far behind men

Women who return to work part-time after having a baby continue to earn less than men for many years afterwards, says a report by the Institute for Fiscal Studies.

?Square Kilometre Array software prototype runs on Chinese supercomputer

A prototype part of the software system to manage data from the Square Kilometre Array telescope has successfully run on the world's second-fastest supercomputer in China.

Lenovo bloats up Android with Microsoft Office and Skype

As part of a patent licensing deal with Microsoft, Lenovo will preinstall Microsoft Office, Skype, and OneDrive on select devices.

Retailers, payments association want banks granted negotiation rights with Apple

Coles, the Australian Payments Clearing Association, and the Australian Retailers Association believe granting Australian banks the right to negotiate with Apple will promote innovation, competition, and greater transparency.

Ramen noodles 'are most valuable US prison commodity', study finds

Ramen noodles have overtaken tobacco to become the most valuable commodity in US prisons, a new study says.

Victorian government on the hunt for a datacentre provider

The Victorian WorkCover Authority and the Transport Accident Commission have gone to tender for a vendor to provide up to two datacentres for the state government agencies.

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